A | B |
alpha-1 | Vascular Smooth Muscle (adventitial layer) |
alpha-2 | Presynaptic Adrenergic Nerve Terminals |
beta-1 | Myocardium |
beta-2 | Vascular Smooth Muscle (luminal) |
M1 | Presynaptic Cholinergic Nerve Terminal |
M2 | Vascular Endothelium |
NN (NG) | Autonomic Ganglia |
alpha-1 | Vasoconstriction |
alpha-2 | Inhibition of Transmitter Release |
beta-1 | Increased Inotropy and Chronotropy |
beta-2 | Vasodilation |
M1 | Inhibition of Transmitter Release |
M2 | Vasodilation (via Nitric Oxide (EDRF)) |
NN (NG) | Impulse Propagation |
Epinephrine | alpha-1, alpha-2, beta-1, beta-2 agonist |
Norepinephrine | alpha-1, alpha-2, beta-1 agonist |
Phenylephrine | alpha-1 agonist |
Isoproterenol | beta-1, beta-2 agonist |
Acetylcholine | M1, M2 agonist |
Hexamethonium (C6) | NN (NG): Antagonist |
Propranolol | beta-1, beta-2 : Antagonist |
Prazosin | alpha-1 Antagonist |
Atropine : receptors | M1, M2 Antagonist (Slightly more M1 than M2) |
alhpha-2 | vascular smooth muscle constriction ( minor effect) |
Presynaptic Cholinergic Nerve Terminal | beta-2 |
inhibition of transmitter release | beta-2 |