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Autonomic Pharmacology : Cardiology

AB
alpha-1Vascular Smooth Muscle (adventitial layer)
alpha-2Presynaptic Adrenergic Nerve Terminals
beta-1Myocardium
beta-2Vascular Smooth Muscle (luminal)
M1Presynaptic Cholinergic Nerve Terminal
M2Vascular Endothelium
NN (NG)Autonomic Ganglia
alpha-1Vasoconstriction
alpha-2Inhibition of Transmitter Release
beta-1Increased Inotropy and Chronotropy
beta-2Vasodilation
M1Inhibition of Transmitter Release
M2Vasodilation (via Nitric Oxide (EDRF))
NN (NG)Impulse Propagation
Epinephrinealpha-1, alpha-2, beta-1, beta-2 agonist
Norepinephrinealpha-1, alpha-2, beta-1 agonist
Phenylephrinealpha-1 agonist
Isoproterenolbeta-1, beta-2 agonist
AcetylcholineM1, M2 agonist
Hexamethonium (C6)NN (NG): Antagonist
Propranololbeta-1, beta-2 : Antagonist
Prazosinalpha-1 Antagonist
Atropine : receptorsM1, M2 Antagonist (Slightly more M1 than M2)
alhpha-2vascular smooth muscle constriction ( minor effect)
Presynaptic Cholinergic Nerve Terminalbeta-2
inhibition of transmitter releasebeta-2



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